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1

Radioligand binding to intact cells as a tool for extended drug screening in a representative physiological context

Vauquelin, Georges, Van Liefde, Isabelle, Swinney, David C.

Journal:

Drug Discovery Today: Technologies

Year:

2015

Language:

english

File:

PDF, 692 KB

english, 2015

2

Human M1-, M2- and M3-muscarinic cholinergic receptors: Binding characteristics of agonists and antagonists

Patrick Vanderheyden, Jean-Pierre Gies, Guy Ebinger, Jacques De Keyser, Yves Landry, Georges Vauquelin

Journal:

Journal of the Neurological Sciences

Year:

1990

Language:

english

File:

PDF, 739 KB

english, 1990

3

Evaluation of bioactive saponins and triterpenoidal aglycons for their binding properties on human endothelin ETA and angiotensin AT1 receptors

C. Caballero-George, P. M. L. Vanderheyden, Y. Okamoto, T. Masaki, Z. Mbwambo, S. Apers, M. P. Gupta, L. Pieters, G. Vauquelin, A. Vlietinck

Journal:

Phytotherapy Research

Year:

2004

Language:

english

File:

PDF, 245 KB

english, 2004

4

Involvement of insulin-regulated aminopeptidase and/or aminopeptidase N in the angiotensin IV-induced effect on dopamine release in the striatum of the rat

Bart Stragier, Heidi Demaegdt, Dimitri De Bundel, Ilse Smolders, Sophie Sarre, Georges Vauquelin, Guy Ebinger, Yvette Michotte, Patrick Vanderheyden

Journal:

Year:

2007

Language:

english

File:

PDF, 649 KB

english, 2007

5

D1 dopamine receptors in human putamen, frontal cortex and calf retina: differences in guanine nucleotide regulation of agonist binding and adenylate cyclase stimulation

Jacques De Keyser, Rudi Dierckx, Patrick Vanderheyden, Guy Ebinger, Georges Vauquelin

Journal:

Year:

1988

Language:

english

File:

PDF, 778 KB

english, 1988

6

Angiotensin II type 1 receptor antagonists: Why do some of them produce insurmountable inhibition?

Patrick M.L Vanderheyden, Frederik L.P Fierens, Georges Vauquelin

Journal:

Biochemical Pharmacology

Year:

2000

Language:

english

File:

PDF, 412 KB

english, 2000

7

Insurmountable AT1 receptor antagonism: the need for different antagonist binding states of the receptor

Georges Vauquelin, Frederik Fierens, Ilse Verheijen, Patrick Vanderheyden

Journal:

Trends in Pharmacological Sciences

Year:

2001

Language:

english

File:

PDF, 35 KB

english, 2001

8

Identification of I1 and I2 Imidazoline Receptors in Striatum Membranes from Different Speciesa

GEORGES VAUQUELIN, JEAN-PAUL DE BACKER, PHILIPPE LADURE, ANJA FLAMEZ

Journal:

Annals of the New York Academy of Sciences

Year:

1999

File:

PDF, 808 KB

1999

9

Corrigendum

Hilde De Vos, Eva Czerwiec, Jean-Paul De Backer, Werner De Potter, Georges Vauquelin

Journal:

European Journal of Pharmacology: Molecular Pharmacology

Year:

1991

Language:

english

File:

PDF, 41 KB

english, 1991

10

Angiotensin AT4 receptor ligand interaction with cystinyl aminopeptidase and aminopeptidase N: [125I]Angiotensin IV only binds to the cystinyl aminopeptidase apo-enzyme

Heidi Demaegdt, Pieter-Jan Lenaerts, Julie Swales, Jean-Paul De Backer, Hilde Laeremans, Minh Tam Le, Ken Kersemans, Lotte K. Vogel, Yvette Michotte, Patrick Vanderheyden, Georges Vauquelin

Journal:

European Journal of Pharmacology

Year:

2006

Language:

english

File:

PDF, 260 KB

english, 2006

11

Non-competitive binding of the nonpeptide antagonist BIBP3226 to rat forebrain neuropeptide Y1 receptors

Patrick M.L Vanderheyden, Isabelle Van Liefde, Jean-Paul De Backer, Georges Vauquelin

Journal:

European Journal of Pharmacology

Year:

1997

Language:

english

File:

PDF, 321 KB

english, 1997

12

(±)Tetrahydroanisocycline and (±)tetrahydropalmatine binding to D1 and D2 dopaminergic receptors in human putamen

Vauquelin, Georges, De Keyser, Jacques, Kanyinda, Banyingela, Vanhaelen, Maurice

Journal:

Neurochemistry International

Year:

1989

Language:

english

File:

PDF, 302 KB

english, 1989

13

[3H]Rauwolscine labels α2-adrenoceptors and 5-HT1A receptors in human cerebral cortex

André Convents, Jacques De Keyser, Jean-Paul De Backer, Georges Vauquelin

Journal:

European Journal of Pharmacology

Year:

1989

Language:

english

File:

PDF, 274 KB

english, 1989

14

On the different experimental manifestations of two-state ‘induced-fit’ binding of drugs to their cellular targets

Vauquelin, Georges, Van Liefde, Isabelle, Swinney, David C

Journal:

British Journal of Pharmacology

Year:

2016

Language:

english

File:

PDF, 2.81 MB

english, 2016

15

Insurmountable AT1 receptor antagonism: fitting models with experimental data

Georges Vauquelin, Frederik FierensIlse, VerheijenPatrick Vanderheyden

Journal:

Trends in Pharmacological Sciences

Year:

2001

Language:

english

File:

PDF, 18 KB

english, 2001

16

Inhibitory Activity on Binding of Specific Ligands to the Human Angiotensin II AT 1 and Endothelin 1 ET A Receptors: Bioactive Benzo[ c ]phenanthridine Alkaloids from the Root of Bocconia frutescens

Caballero-George, Catherina, Vanderheyden, Patrick M., Apers, Sandra, Van den Heuvel, Hilde, Solis, Pablo N., Gupta, Mahabir P., Claeys, Magda, Pieters, Luc, Vauquelin, Georges, Vlietinck, Arnold J.

Journal:

Year:

2002

Language:

english

File:

PDF, 237 KB

english, 2002

17

Involvement of the AT1 receptor subtype in the effects of angiotensin IV and LVV-haemorphin 7 on hippocampal neurotransmitter levels and spatial working memory

Dimitri De Bundel, Heidi Demaegdt, Tony Lahoutte, Vicky Caveliers, Ken Kersemans, Ann-Gaelle Ceulemans, Georges Vauquelin, Ralph Clinckers, Patrick Vanderheyden, Yvette Michotte, Ilse Smolders

Journal:

Journal of Neurochemistry

Year:

2010

Language:

english

File:

PDF, 942 KB

english, 2010

18

Dopamine and Iron Induce Apoptosis in PC12 Cells

Carlos Velez-Pardo, Marlene Jimenez Del Rio, Hendrik Verschueren, Guy Ebinger, Georges Vauquelin

Journal:

Basic & Clinical Pharmacology & Toxicology

Year:

1997

Language:

english

File:

PDF, 1.19 MB

english, 1997

19

Cys2,7EtαCGRP is a potent agonist for CGRP1 receptors in SK-N-MC cells

Christina Nodin, Georges Vauquelin, Bengt von Mentzer

Journal:

Biochemical Pharmacology

Year:

2005

Language:

english

File:

PDF, 179 KB

english, 2005

20

Dual effect of N-ethylmaleimide on agonist-mediated conformational changes of β-adrenergic receptors

Claudine Andre, Georges Vauquelin, Yvonne Severne, Jean-Paul De Backer, A. Donny Strosberg

Journal:

Biochemical Pharmacology

Year:

1982

Language:

english

File:

PDF, 518 KB

english, 1982

21

Isoproterenol and selective agonists stimulate similar atypical β-adrenoceptors in rat adipocytes

Isabelle Van Liefde, Anne van Witzenburg, Georges Vauquelin

Journal:

Biochemical Pharmacology

Year:

1993

Language:

english

File:

PDF, 398 KB

english, 1993

22

Serotonin Binding Proteins: An In Vitro Model System for Monoamine-related Neurotoxicity

GEORGES VAUQUELIN, MARLENE JIMENEZ DEL RIO, CARLOS VELEZ PARDO

Journal:

Annals of the New York Academy of Sciences

Year:

1994

Language:

english

File:

PDF, 712 KB

english, 1994

23

Simplified models for heterobivalent ligand binding: when are they applicable and which are the factors that affect their target residence time

Georges Vauquelin

Journal:

Naunyn-Schmiedeberg's Archives of Pharmacology

Year:

2013

Language:

english

File:

PDF, 567 KB

english, 2013

24

On the ‘micro’-pharmacodynamic and pharmacokinetic mechanisms that contribute to long-lasting drug action

Vauquelin, Georges

Journal:

Expert Opinion on Drug Discovery

Year:

2015

Language:

english

File:

PDF, 797 KB

english, 2015

25

Long-lasting angiotensin type 1 receptor binding and protection by candesartan: comparison with other biphenyl-tetrazole sartans

Vauquelin, Georges, Fierens, Frederik, Liefde, Isabelle Van

Journal:

Journal of Hypertension

Year:

2006

Language:

english

File:

PDF, 339 KB

english, 2006

26

D2 Dopamine Receptors in Calf Globus Pallidus: Agonist High- and Low-Affinity Sites Not Regulated by Guanine Nucleotide

Jacques De Keyser, Jean-Paul De Backer, André Convents, Guy Ebinger, Georges Vauquelin

Journal:

Journal of Neurochemistry

Year:

1985

Language:

english

File:

PDF, 330 KB

english, 1985

27

Effect of saponin and filipin on antagonist binding to AT1 receptors in intact cells

Ilse Verheijen, Dieter Tourlousse, Patrick M.L Vanderheyden, Jean-Paul De Backer, Georges Vauquelin

Journal:

Biochemical Pharmacology

Year:

2004

Language:

english

File:

PDF, 196 KB

english, 2004

28

Agonist mediated conformational changes of solubilized calf forebrain muscarinic acetylcholine receptors

Patrick Vanderheyden, Claudine Andre, Jean-Paul de Backer, Georges Vauquelin

Journal:

Biochemical Pharmacology

Year:

1984

Language:

english

File:

PDF, 634 KB

english, 1984

29

Human neuropeptide YY1 receptors exert unequal control of the extracellular acidification rate in different cell lines

Isabelle Van Liefde, Patrick M.L Vanderheyden, Norbert Fraeyman, Jean-Paul De Backer, Georges Vauquelin

Journal:

European Journal of Pharmacology

Year:

1998

Language:

english

File:

PDF, 299 KB

english, 1998

30

Link between a high kon for drug binding and a fast clinical action: to be or not to be ?

Vauquelin, Georges

Journal:

Year:

2018

Language:

english

File:

PDF, 1.65 MB

english, 2018

31

Clozapine, atypical antipsychotics, and the benefits of fast-off D2dopamine receptor antagonism

Georges Vauquelin, Sophie Bostoen, Patrick Vanderheyden, Philip Seeman

Journal:

Naunyn-Schmiedeberg's Archives of Pharmacology

Year:

2012

Language:

english

File:

PDF, 981 KB

english, 2012

32

Ligand binding and functional properties of human angiotensin AT1 receptors in transiently and stably expressed CHO-K1 cells

Minh Tam Le, Jean-Paul De Backer, László Hunyady, Patrick M.L. Vanderheyden, Georges Vauquelin

Journal:

European Journal of Pharmacology

Year:

2005

Language:

english

File:

PDF, 467 KB

english, 2005

33

Corticotropin-releasing factor receptors induce calcium mobilization through cross-talk with Gq-coupled receptors

Eric Gutknecht, Georges Vauquelin, Frank M. Dautzenberg

Journal:

European Journal of Pharmacology

Year:

2010

Language:

english

File:

PDF, 1.10 MB

english, 2010

34

Antagonist interaction with endogenous AT1 receptors in human cell lines

Ilse Verheijen, Patrick M.L Vanderheyden, Jean-Paul De Backer, Serge Bottari, Georges Vauquelin

Journal:

Biochemical Pharmacology

Year:

2002

Language:

english

File:

PDF, 156 KB

english, 2002

35

Models and methods for studying insurmountable antagonism

Georges Vauquelin, Isabelle Van Liefde, Patrick Vanderheyden

Journal:

Trends in Pharmacological Sciences

Year:

2002

Language:

english

File:

PDF, 64 KB

english, 2002

36

125I-Tyr0-hCRH Labelling characteristics of corticotropin-releasing hormone receptors: differences between normal and adenomatous corticotrophs

Roger Abs, Gerda Smets, Georges Vauquelin, Johan Verhelst, Charles Mahler, Jan Verlooy, Achille Stevenaert, Luc Wouters, Marcel Borgers, Albert Beckers

Journal:

Neurochemistry International

Year:

1997

Language:

english

File:

PDF, 573 KB

english, 1997

37

Identification and characterization of α2-adrenergic receptors in human myometrium by [3H]rauwolscine binding

Bottari, Serge P., Vokaer, Alain, Kaivez, Etienne, Lescrainier, Jean Paul, Vauquelin, Georges

Journal:

American Journal of Obstetrics and Gynecology

Year:

1983

Language:

english

File:

PDF, 546 KB

english, 1983

38

Conformational constraints in angiotensin IV to probe the role of Tyr2, Pro5 and Phe6

Aneta Lukaszuk, Heidi Demaegdt, Isabelle Van den Eynde, Patrick Vanderheyden, Georges Vauquelin, Dirk Tourwé

Journal:

Journal of Peptide Science

Year:

2011

Language:

english

File:

PDF, 279 KB

english, 2011

39

Antagonist-D2S-dopamine receptors interactions in intact Chinese recombinant ovary cells

Ann Packeu, Tim Béghin, Jean-Paul De Backer, Georges Vauquelin

Journal:

Fundamental & Clinical Pharmacology

Year:

2010

Language:

english

File:

PDF, 250 KB

english, 2010

40

[3H]GBR 12935 Binding to Dopamine Uptake Sites in the Human Brain

Jacques De Keyser, Jean-Paul De Backer, Guy Ebinger, Georges Vauquelin

Journal:

Journal of Neurochemistry

Year:

1989

Language:

english

File:

PDF, 1011 KB

english, 1989

41

Radioligand dissociation measurements: potential interference of rebinding and allosteric mechanisms and physiological relevance of the biological model systems

Vauquelin, Georges, Van Liefde, Isabelle

Journal:

Expert Opinion on Drug Discovery

Year:

2012

Language:

english

File:

PDF, 406 KB

english, 2012

42

Serotonin-binding proteins in the bovine cerebral cortex: interaction with serotonin and catecholamines

Marlene Jimenez Del Rio, Jef Pinxteren, Werner Do Potter, Guy Ebinger, Georges Vauquelin

Journal:

European Journal of Pharmacology: Molecular Pharmacology

Year:

1992

Language:

english

File:

PDF, 1.01 MB

english, 1992

43

Distinction between Two Subpopulations of β1-Adrenergic Receptors in Human Adipose Cells

Bo JACOBSSON, Georges VAUQUELIN, Christian WESSLAU, Ulf SMITH, A. Donny STROSBERG

Journal:

Year:

1981

Language:

english

File:

PDF, 626 KB

english, 1981

44

Agonist-Mediated Conformational Changes of Muscarinic Receptors in Rat Brain

Georges VAUQUELIN, Claudine ANDRÉ, Jean-Paul DE BACKER, Pierre LADURON, A. Donny STROSBERG

Journal:

Year:

1982

Language:

english

File:

PDF, 870 KB

english, 1982

45

Endogenous noradrenaline masks beta-adrenergic receptors in rat heart membranes via tight agonist binding

Viveca Nerme, Yvonne Severne, Tommy Abrahamsson, Georges Vauquelin

Journal:

Biochemical Pharmacology

Year:

1985

Language:

english

File:

PDF, 593 KB

english, 1985

46

Agonist/N-ethylmaleimide mediated inactivation of β-adrenergic receptors: Molecular aspects

Yvonne Severne, Claire Wemers, Georges Vauquelin

Journal:

Biochemical Pharmacology

Year:

1985

Language:

english

File:

PDF, 582 KB

english, 1985

47

Binding of “AT4 receptor” ligands to insulin regulated aminopeptidase (IRAP) in intact Chinese hamster ovary cells

Heidi Demaegdt, Paul Gard, Jean-Paul De Backer, Aneta Lukaszuk, Erzsébet Szemenyei, Géza Tóth, Dirk Tourwé, Georges Vauquelin

Journal:

Molecular and Cellular Endocrinology

Year:

2011

Language:

english

File:

PDF, 1009 KB

english, 2011

48

Agonist induction and conformational selection during activation of a G-protein-coupled receptor

László Hunyady, Georges Vauquelin, Patrick Vanderheyden

Journal:

Trends in Pharmacological Sciences

Year:

2003

Language:

english

File:

PDF, 403 KB

english, 2003

49

Identification of α2 adrenergic receptors in human frontal cortex membranes by binding of [3H]RX 821002, the 2-methoxy analog of [3H]idazoxan

Vauquelin, Georges, De Vos, Hilde, De Backer, Jean-Paul, Ebinger, Guy

Journal:

Neurochemistry International

Year:

1990

Language:

english

File:

PDF, 798 KB

english, 1990

50

Metal ion modulation of cystinyl aminopeptidase

Laeremans, Hilde, Demaegdt, Heidi, De Backer, Jean-Paul, Le, Minh T., Kersemans, Veerle, Michotte, Yvette, Vauquelin, Georges, Vanderheyden, Patrick M. L.

Journal:

Biochemical Journal

Year:

2005

Language:

english

File:

PDF, 380 KB

english, 2005

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